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194 Inhibitors against Fungal Cell Wall Remodeling Enzymes
ChemMedChem
2018, 13, 128-132. DOI: 10.1002/cmdc.201700720
Thumbnail image of graphical abstract
193 (+)-Methyl (1R,2S)-2-{[4-(4-Chlorophenyl)-4-hydroxypiperidin-1-yl]methyl}-1-phenylcyclopropanecarboxylate [(+)-MR200] Derivatives as Potent and Selective Sigma Receptor Ligands: Stereochemistry and Pharmacological Properties
J. Med. Chem.
2018, 61, 372-384. DOI: 10.1021/acs.jmedchem.7b01584
Figure
192 Exploratory spectroscopic and computational studies of the anion binding properties of methyl hyocholate in organic solvent
Org. Chem. Front.
2018, 6, 0000-0000. DOI: 10.1039/C7QO00858A
Graphical abstract: Synergistic catalysis: enantioselective cyclopropanation of alkylidene benzoxazoles by Pd(ii) and secondary amine catalysis. Scope, limitations and mechanistic insight
191 Introducing topology to assess the synchronicity of organic reactions. Dual reactivity of oximes with alkenes as a case study
Org. Chem. Front.
2017, 4, 1541-1554. DOI: /10.1039/C7QO00233E
Graphical abstract: Introducing topology to assess the synchronicity of organic reactions. Dual reactivity of oximes with alkenes as a case study
190 One-Pot Synthesis of Functionalized Carbazoles via a CAN-Catalyzed Multicomponent Process Comprising a C–H Activation Step
J. Org. Chem.
2017, 82, 7493-7502. DOI: 10.1021/acs.joc.7b01199
Abstract Image
189 Nitrones and nucleobase-containing spiro-isoxazolidines derived from isatin and indanone: solvent-free microwave-assisted stereoselective synthesis and theoretical calculations
RSC Adv.
2017, 7, 48980-48988. DOI: 10.1039/C7RA09995A
Graphical abstract: Nitrones and nucleobase-containing spiro-isoxazolidines derived from isatin and indanone: solvent-free microwave-assisted stereoselective synthesis and theoretical calculations
188

Exploratory spectroscopic and computational studies of the anion binding properties of methyl hyocholate in organic solvent
Tetrahedron
2017, 73, 1698-1704. DOI: 10.1016/j.tet.2017.02.015

187 BET & ELF Quantum Topological Analysis of Neutral 2-Aza-Cope Rearrangement of γ-Alkenyl Nitrones
Molecules
2017, 22, 1371-1383. DOI: 10.3390/molecules22081371
186

The small molecule luteolin inhibits N-acetyl-α-galactosaminyltransferases and reduces mucin-type O-glycosylation of amyloid precursor protein
J. Biol. Chem.
2017, 292, 21304-21319. DOI: 10.1074/jbc.M117.814202

Figure 3.

185 A Case Study of Thiourea-Assisted Iminium Formation by Hydroxyl Anion Binding: Kinetic, Spectroscopic and Computational Evidences
Adv. Synth. Catal.
2017, 359, 4122-4128. DOI: 10.1002/adsc.201700986
184 Organocatalytic Enantioselective Synthesis of Trifluoromethyl-Containing Tetralin Derivatives by Sequential (Hetero)Michael Reaction–Intramolecular Nitrone Cycloaddition
Adv. Synth. Catal.
2017, 359, 3752-3764. DOI: 10.1002/adsc.201700975
183 Racemic Hemiacetals as Oxygen-Centered Pronucleophiles Triggering Cascade 1,4-Addition/Michael Reaction through Dynamic Kinetic Resolution under Iminium catalysis. Reaction Development and Mechanistic Insights
Chem. Sci.
2017, 8, 2904-2913. DOI: 10.1039/C7SC00009J
182 Regioselectivity Change in the Organocatalytic Enantioselective (3+2) Cycloaddition with Nitrones Through Cooperative H-Bonding Catalysis/Iminium Activation
Chem. Eur. J.
2017, 23, 2764-2768. DOI: 10.1002@chem.201605350

181 A Molecular Electron Density Theory Study of the [3+2] Cycloaddition Reaction of Nitrones with Ketenes
Org. Biol. Chem.
2017, 15, 1525-1534. DOI: 10.1039/C6OB02768G
180 Pivotal Neighbouring Group Participation in Substitution vs Elimination Reactions: Computational Evidence for Ion Pairs in the Thionation of Alcohols with Lawesson's Reagent
Eur. J. Org. Chem. 2017, 1952-1960 DOI: 10.1002/ejoc.201700127

179

Synthesis of Amino Acid-Nucleoside Conjugates, Ghirardello, M.; Delso, I.; Tejero, T.; Merino, P.
Asian
J. Org. Chem.. 2016, 1525-1534. DOI: 10.1002/ajoc.201600497

178

Computational Mechanistic Study of Thionation of Carbonyl Compounds with Lawesson's Reagent, Juste-Navarro, V.; Delso, I.; Tejero, T.; Merino, P.
J. Org. Chem.. 2016, 81, 7733-7740. DOI: 10.1021/acs.joc.6b01420

177

Azomethine Ylides from Nitrones: Using Catalytic n-BuLi for the Totally Stereoselective Synthesis of trans-2-Alkyl-3-Oxazolines, Juste-Navarro, V.; Delso, I.; Tejero, T.; Merino, P.
Chem. Eur. J.
2016, 22, 11527-11532. DOI: 10.1002/chem.201602159. Cover: DOI: 10.1002/chem.201602827.
Cover Profile: DOI: 10.1002/chem.201602894

176

Glycomimetics Targeting Glycosyltransferases: Synthetic, Computational and Structural Studies of Less-Polar Conjugates, Ghirardello, M.; de las Rivas, M.; Lacetera, A.; Delso, I.; Lira-Navarrete, E.; Tejero, T.; Martin-Santamaria, S.; Hurtado-Guerrero, R.; Merino, P.
Chem. Eur. J.
2016, 22, 7215-7224. DOI: 10.1002/chem.201600467

175

Mechanistic Insights in the Mode of Action of Bifunctional Pyrrolidine-Squaramide-derived Organocatalysts, Roca-López, D.; Uria, U.; Reyes, E.; Carrillo, L.; Jørgensen, K. A.; Vicario, J. L.; Merino, P.
Chem. Eur. J. 2016, 22, 884-889. DOI: 10.1002/chem.201504705

174

Revisiting Oxime-Nitrone Tautomerism. Evidences of Nitrone Tautomer Participation in Oxime Nucleophilic Addition Reactions, Roca-López, D.; Darù, A.; Tejero, T.; Merino, P.
RSC Adv.
2016, 6, 22161-22173. DOI: 10.1039/C6RA02638A

173

Rapid, Efficient and Solvent Free MW Mediated Synthesis of Aldo- and Ketonitrones, Maiuolo, L.; Nino, A. D.; Merino, P.; Russo, B.; Stabile, G.; Nardi, M.; D’Agostino, N.; Bernardi, T. Arabian J. Chem. 2016, 9, 25-31. DOI: 10.1016/j.arabjc.2015.01.015

172

Stereoselective Ethynylation and Propargylation of Chiral Cyclic Nitrones. Application to the Synthesis of Glycomimetics, García-Viñuales, S.; Delso, I.; Merino, P.; Tejero, T. Synthesis 2016, DOI: 10.1055/s-0035-1562500

171

Rational design of glycomimetic compounds targeting the Saccharomyces cerevisae transglycosylase Gas2, Delso, I.; Valero-González, J.; Marca, E.; Tejero, T.; Hurtado-Guerrero, R.; Merino, P. Chem. Biol. Drug Design 2016, 87, 163-170. DOI: 10.1111/cbdd.12650

170

Revealing Stepwise Mechanisms in Dipolar Cycloaddition Reactions: Computational Study of the Reaction between Nitrones and Isocyanates, Daru, A.; Roca-López, D.; Tejero, T.; Merino, P. J. Org. Chem. 2016, 81, 673-680. DOI: 10.1021/acs.joc.5b02645

169

Mechanism Switch in Mannich-type Reactions. ELF and NCI Topological Analyses of the Reaction between Nitrones and Lithium Enolates, Roca-López, D.; Polo, V.; Tejero, T.; Merino, P. Eur. J. Org. Chem. 2015, 4143-4152.

168

Understanding Bond Formation in Polar One-Step Reactions. Topological analyses of the Reaction between Nitrones and Lithium Ynolates, Roca-López, D.; Polo, V.; Tejero, T.; Merino, P. J. Org. Chem. 2015, 80, 4076-4083.

167

New Efficient Organocatalyst Supported on Simple Ionic Liquid as Recoverable System for Asymmetric Diels-Alder Reaction in Presence of Water, Nino, A. D.; Maiuolo, L.; Merino, P.; Nardia, M.; Procopio, A.; Roca-López, D.; Russo, B. ChemCatChem 2015, 7, 830-835.

166

A Natural Ternary Complex Trapped in Crystal Reveals the Catalytic Mechanism of a Retaining Glycosyltransferase, Albesa-Jové, D.; Mendoza, M. F.; Rodrigo-Unzueta, A.; Gomollón-Bel, F.; Cifuente, J.; Urresti, S.; Comino, N.; Gómez, H.; Romero-García, J.; Lluch, J. M.; Sancho-Vaello, E.; Biarnés, X.; Planas, A.; Merino, P.; Masgrau, L.; Guerin, M. E. Angew. Chem. Int. Ed. 2015, 54, 9898-9902.

165

DFT Investigation of the Mechanism of E/Z Isomerization of Nitrones, Roca-Lopez, D.; Tejero, T.; Merino, P. J. Org. Chem. 2014, 79, 8358-8365.

164

[2n2π + 2n2π] Cycloadditions: An alternative to forbidden [4π + 4π] processes. The Case of Nitrones Dimerizations, Roca-López, D.; Tejero, T.; Caramella, P.; Merino, P. Org. Biomol. Chem. 2014, 12, 517-525.

163

Friedel-Crafts alkylation mechanism using aminoindanol derived thiourea catalyst, Roca-López, D.; Marqués-López, E.; Alcaine, A.; Merino, P.; Herrera, R. P. Org. Biomol. Chem. 2014, 12, 4503-4510.

162

Theoretical Elucidation of the Mechanism of the Cycloaddition between Nitrone Ylides and Electron-deficient Alkenes, Merino, P.; Tejero, T.; Diez Martinez, A. J. Org. Chem. 2014, 79, 2189-2202.

161

Highly Diastereoselective 1,3-Dipolar Cycloadditions of Chiral Non-Racemic Nitrones to 1,2-Diaza-1,3-dienes: An Experimental and Computational Investigation, Majer, R.; Konechnaya, O.; Delso, I.; Tejero, T.; Attanasi, O. A.; Santeusanio, S.; Merino, P. Org. Biomol. Chem. 2014, 12, 8888-8901.

160

Stereoselective 1,3-dipolar cycloadditions of nitrones derived from amino acids. Asymmetric synthesis of N-(alkoxycarbonylmethyl)-3-hydroxypyrrolidin-2-ones, Merino, P.; Greco, G.; Tejero, T.; Hurtado-Guerrero, R.; Matute, R.; Chiacchio, U.; Corsaro, A.; Pistara, V.; Romeo, R. Tetrahedron 2013, 69, 9381-9390.

159

Synthesis of O- and C-glycosides derived from β-(1,3)-D-glucans Marca, E.; Valero-Gonzalez, J.; Delso, I.; Tejero, T.; Hurtado-Guerrero, R.; Merino, P. Carbohydr. Res. 2013, 382, 9-18.

158

The High Selectivity of the Cp2ZrHCl Reducing Agent for Imides: A Combined Experimental and Theoretical Study on γ-Lactam and Isoxazolidinone Derivatives, Lanza, G.; Chiacchio, M. A.; Giofre, S. V.; Romeo, R.; Merino, P. Eur. J. Org. Chem. 2013, 2013, 95-104.

157

Evasive Neutral 2-Aza-Cope Rearrangements. Kinetic and Computational Studies with Cyclic Nitrones, Delso, I.; Melicchio, A.; Isasi, A.; Tejero, T.; Merino, P. Eur. J. Org. Chem. 2013, 2013, 5721-5730.

156

Truncated Reverse Isoxazolidinyl Nucleosides: A New Class of Allosteric HIV-1 Reverse Transcriptase Inhibitors, Romeo, R.; Giofrè, S. V.; Macchi, B.; Balestrieri, E.; Mastino, A.; Merino, P.; Carnovale, C.; Romeo, G.; Chiacchio, U. ChemMedChem 2012, 7, 565-569.

155

Highly stereoselective synthesis of imino-C-di- and trisaccharides as hydrolytically stable glycomimetics, Marca, E.; Delso, I.; Tejero, T.; Merino, P. Tetrahedron 2012, 68, 6674-6687.

154

Dual reactivity of O-α-allenyl esters under palladium(0) catalysis: From carbopalladation/allylic alkylation domino sequence to decarboxylative allenylation, Kammerer-Pentier, C.; Diez Martinez, A.; Oble, J.; Prestat, G.; Merino, P.; Poli, G. J. Organomet. Chem. 2012, 714, 53-59.

153

Stereoselective Hydride Transfer by Aryl-Alcohol Oxidase, a Member of the GMC Superfamily, Hernandez-Ortega, A.; Ferreira, P.; Merino, P.; Medina, M.; Guallar, V.; Martinez, A. T. ChemBioChem 2012, 13, 427-435.

152

Water-compatible one-pot organocatalytic asymmetric synthesis of cyclic nitrones. Application in intramolecular 1,3-dipolar cycloadditions, Sadaba, D.; Delso, I.; Tejero, T.; Merino, P. Tetrahedron Lett. 2011, 52, 5976-5979.

151

Organocatalyzed Michael addition reaction by novel (2R,3aS,7aS)-octahydroindole-2-carboxylic acid, a new fused proline, Roca-Lopez, D.; Merino, P.; Sayago, F. J.; Cativiela, C.; Herrera, R. P. Synlett 2011, 249-253.

150

Nitrone ylides: Two possible 1,3-dipolar cycloadditions but only one stepwise formation of all-cis 2,4,5-trisubstituted N-hydroxypyrrolidines, Merino, P.; Tejero, T.; Diez-Martinez, A.; Gultekin, Z. Eur. J. Org. Chem. 2011, 6567-6573.

149

High-yield synthesis of pyrrolidinyl PNA monomers, Merino, P.; Greco, G.; Tejero, T.; Corsaro, A.; Chiacchio, U.; Pistara, V.; Romeo, G. Tetrahedron Lett. 2011, 52, 6003-6006.

148

Structural insights into the mechanism of Protein O-fucosylation, Lira-Navarrete, E.; Valero-Gonzalez, J.; Villanueva, R.; Martinez-Julvez, M.; Tejero, T.; Merino, P.; Panjikar, S.; Hurtado-Guerrero, R. PLoS One 2011, 9, e25365 (14 pages).

147

Sequential nucleophilic addition/intramolecular cycloaddition to chiral nonracemic cyclic nitrones: A highly stereoselective approach to polyhydroxynortropane alkaloids, Delso, I.; Tejero, T.; Goti, A.; Merino, P. J. Org. Chem. 2011, 76, 4139-4143.

146

Thiourea catalyzed organocatalytic enantioselective Michael addition of diphenyl phosphite to nitroalkenes, Alcaine, A.; Marques-Lopez, E.; Merino, P.; Tejero, T.; Herrera, R. P. Org. Biomol. Chem. 2011, 9, 2777-2783.

145

Asymmetric organocatalytic synthesis of γ-nitrocarbonyl compounds through Michael and Domino reactions, Roca-Lopez, D.; Sadaba, D.; Delso, I.; Herrera, R. P.; Tejero, T.; Merino, P. Tetrahedron Asymmetry 2010, 21, 2561-2601.

144

Expanding the limits of organoboron chemistry: Synthesis of functionalized arylboronates, Merino, P.; Tejero, T. Angew. Chem. Int. Ed. 2010, 49, 7164-7165.

143

Enantioselective organocatalytic Diels-Alder reactions, Merino, P.; Marques-Lopez, E.; Tejero, T.; Herrera, R. P. Synthesis 2010, 1-26.

142

Experimental and theoretical studies on Mannich-type reactions of chiral non-racemic N-(benzyloxyethyl) nitrones, Diez-Martinez, A.; Tejero, T.; Merino, P. Tetrahedron Asymmetry 2010, 21, 2934-2943.

141

Synthesis of N-(benzyloxyethyl)- and N-(alkoxycarbonylmethyl)nitrones, Diez-Martinez, A.; Gultekin, Z.; Delso, I.; Tejero, T.; Merino, P. Synthesis 2010, 678-688.

140

Synthesis of D-arabinose-derived polyhydroxylated pyrrolidine, indolizidine and pyrrolizidine alkaloids. Total synthesis of hyacinthacine A2, Delso, I.; Tejero, T.; Goti, A.; Merino, P. Tetrahedron 2010, 66, 1220-1227.

139

Tunable Diastereoselection of Biased Rigid Systems by Lewis Acid Induced Conformational Effects: A Rationalization of the Vinylation of Cyclic Nitrones En Route to Polyhydroxylated Pyrrolidines, Delso, I.; Marca, E.; Mannucci, V.; Tejero, T.; Goti, A.; Merino, P. Chem. Eur. J. 2010, 16, 9910-9919.

138

Organocatalyzed Strecker reactions, Merino, P.; Marques-Lopez, E.; Tejero, T.; Herrera, R. P. Tetrahedron 2009, 65, 1219-1234.

137

Intramolecular 1,3-dipolar cycloaddition of N-alkenyl nitrones en route to glycosyl piperidines, Marca, E.; Delso, I.; Tejero, T.; Vazquez, J. T.; Dorta, R. L.; Merino, P. Tetrahedron Lett. 2009, 50, 7152-7155.

136

Stereoselective Synthesis and Biological Evaluations of Novel 3'-Deoxy-4'-azaribonucleosides as Inhibitors of Hepatitis C Virus RNA Replication, Chiacchio, U.; Borrello, L.; Crispino, L.; Rescifina, A.; Merino, P.; Macchi, B.; Balestrieri, E.; Mastino, A.; Piperno, A.; Romeo, G. Journal of Medicinal Chemistry 2009, 52, 4054-4057.

135

Catalytic enantioselective hydrophosphonylation of aldehydes and imines, Merino, P.; Marques-Lopez, E.; Herrera, R. P. Advanced Synthesis & Catalysis 2008, 350, 1195-1208.

134

Exploring nitrone chemistry: towards the enantiodivergent synthesis of 6-substituted 4-hydroxypipecolic acid derivatives, Merino, P.; Mannucci, V.; Tejero, T. Eur. J. Org. Chem. 2008, 3943-3959.

133

Nucleophilic additions to cyclic nitrones en route to iminocyclitols - total syntheses of DMDP, 6-deoxy-DMDP, DAB-1, CYB-3, nectrisine, and radicamine B, Merino, P.; Delso, I.; Tejero, T.; Cardona, F.; Marradi, M.; Faggi, E.; Parmeggiani, C.; Goti, A. Eur. J. Org. Chem. 2008, 2929-2947.

132

3-(Aminomethyl)-2-(carboxymethyl)isoxazolidinyl nucleosides: building blocks for peptide nucleic acid analogues, Merino, P.; Tejero, T.; Mates, J.; Chiacchio, U.; Corsaro, A.; Romeo, G. Tetrahedron Asymmetry 2007, 18, 1517-1520.

131

Hydroxylamine oxygen as nucleophile in palladium(0)- and palladium(II)-catalyzed allylic alkylation: a novel access to isoxazolidines, Merino, P.; Tejero, T.; Mannucci, V.; Prestat, G.; Madec, D.; Poli, G. Synlett 2007, 944-948.

130

Experimental and theoretical evidences of 2-aza-Cope rearrangement of nitrones, Merino, P.; Tejero, T.; Mannucci, V. Tetrahedron Lett. 2007, 48, 3385-3388.

129

A DFT study on the 1,3-dipolar cycloaddition reactions of C-(hetaryl) nitrones with methyl acrylate and vinyl acetate, Merino, P.; Tejero, T.; Chiacchio, U.; Romeo, G.; Rescifina, A. Tetrahedron 2007, 63, 1448-1458.

128

Nucleophilic additions and redox reactions of polyhydroxypyrroline N-oxides on the way to pyrrolidine alkaloids: total synthesis of radicamine B, Merino, P.; Delso, I.; Tejero, T.; Cardona, F.; Goti, A. Synlett 2007, 2651-2654.

127

Stereoselective synthesis of pyrrolidinyl glycines from nitrones: complementarity of nucleophilic addition and 1,3-dipolar cycloaddition, Merino, P.; Padar, P.; Delso, I.; Thirumalaikumar, M.; Tejero, T.; Kovacs, L. Tetrahedron Lett. 2006, 47, 5013-5016.

126

Enantiodivergent synthesis of D- and L-erythro-sphingosines through Mannich-type reactions of N-benzyl-2,3-O-isopropylidene-D-glyceraldehyde nitrone, Merino, P.; Jimenez, P.; Tejero, T. J. Org. Chem. 2006, 71, 4685-4688.

125

High stereocontrol in the allylation of chiral non-racemic a-alkoxy and a-amino nitrones, Merino, P.; Delso, I.; Mannucci, V.; Tejero, T. Tetrahedron Lett. 2006, 47, 3311-3314.

124

A DFT study of the molecular mechanisms of the nucleophilic addition of ester-derived lithium enolates and silyl ketene acetals to nitrones: effects of the Lewis acid catalyst, Domingo, L. R.; Arno, M.; Merino, P.; Tejero, T. Eur. J. Org. Chem. 2006, 3464-3472.

123

An efficient approach to enantiomeric isoxazolidinyl analogs of tiazofurin based on nitrone cycloadditions, Merino, P.; Tejero, T.; Unzurrunzaga, F. J.; Franco, S.; Chiacchio, U.; Saita, M. G.; Iannazzo, D.; Piperno, A.; Romeo, G. Tetrahedron: Asymmetry 2005, 16, 3865-3876.

122

Nucleophilic additions of lithiated allylphenylsulfone to nitrones: experimental and theoretical investigations, Merino, P.; Mannucci, V.; Tejero, T. Tetrahedron 2005, 61, 3335-3347.

121

Effect of additional chiral ligands in catalytic enantioselective Mannich-type reactions with nitrones, Merino, P.; Franco, S.; Jimenez, P.; Tejero, T.; Chiacchio, M. A. Lett. Org. Chem. 2005, 2, 302-305.

120

Straightforward synthesis of enantiopure 2-aminomethyl and 2-hydroxymethyl pyrrolidines with complete stereocontrol, Marradi, M.; Cicchi, S.; Ignacio Delso, J.; Rosi, L.; Tejero, T.; Merino, P.; Goti, A. Tetrahedron Lett. 2005, 46, 1287-1290.

119

Zinc(II) Triflate-Controlled 1,3-Dipolar Cycloadditions of C-(2-Thiazolyl)nitrones: Application to the Synthesis of a Novel Isoxazolidinyl Analog of Tiazofurin, Chiacchio, U.; Rescifina, A.; Saita, M. G.; Iannazzo, D.; Romeo, G.; Mates, J. A.; Tejero, T.; Merino, P. J. Org. Chem. 2005, 70, 8991-9001.

118

Enantioselective 1,3-Dipolar Cycloaddition of Nitrones to Methacrolein Catalyzed by (h5-C5Me5)M{(R)-Prophos} Containing Complexes (M = Rh, Ir; (R)-Prophos = 1,2-bis(Diphenylphosphino)propane): On the Origin of the Enantioselectivity, Carmona, D.; Lamata, M. P.; Viguri, F.; Rodriguez, R.; Oro, L. A.; Lahoz, F. J.; Balana, A. I.; Tejero, T.; Merino, P. J. Am. Chem. Soc. 2005, 127, 13386-13398.

117

New Concise Total Synthesis of (+)-Lentiginosine and Some Structural Analogues, Cardona, F.; Moreno, G.; Guarna, F.; Vogel, P.; Schuetz, C.; Merino, P.; Goti, A. J. Org. Chem. 2005, 70, 6552-6555.

116

Diastereo- and enantioselective synthesis of 1’-C-branched N,O-nucleosides, Saita, M. G.; Chiacchio, U.; Iannazzo, D.; Corsaro, A.; Merino, P.; Piperno, A.; Previtera, T.; Rescifina, A.; Romeo, G.; Romeo, R. Nucleosides, Nucleotides & Nucleic Acids 2004, 23, 739-742.

115

Organocatalyzed asymmetric alpha-aminoxylation of aldehydes and ketones--an efficient access to enantiomerically pure alpha-hydroxycarbonyl compounds, diols, and even amino alcohols, Merino, P.; Tejero, T. Angew. Chem. Int. Ed. 2004, 43, 2995-2997.

114

Fully stereoselective nucleophilic addition to a novel chiral pyrroline N-oxide: total syntheses of (2S,3R)-3-hydroxy-3-methylproline and its (2R)-epimer, Merino, P.; Revuelta, J.; Tejero, T.; Cicchi, S.; Goti, A. Eur. J. Org. Chem. 2004, 776-782.

113

Nucleophilic additions of chiral non-racemic enolates to N-benzyl-C-(alkoxymethyl) nitrones, Merino, P.; Franco, S.; Mates, J. A.; Merchan, F. L.; Romero, P.; Tejero, T.; Uriel, S.; Matute, R. Arkivoc 2004, 48-58.

112

Diastereoselective synthesis of homo-N,O-nucleosides, Chiacchio, U.; Genovese, F.; Iannazzo, D.; Librando, V.; Merino, P.; Rescifina, A.; Romeo, R.; Procopio, A.; Romeo, G. Tetrahedron 2004, 60, 441-448.

111

The Complete Characterization of a Rhodium Lewis Acid-Dipolarophile Complex as an Intermediate for the Enantioselective Catalytic 1,3-Dipolar Cycloaddition of C,N-Diphenylnitrone to Methacrolein, Carmona, D.; Lamata, M. P.; Viguri, F.; Rodriguez, R.; Oro, L. A.; Balana, A. I.; Lahoz, F. J.; Tejero, T.; Merino, P.; Franco, S.; Montesa, I. J. Am. Chem. Soc. 2004, 126, 2716-2717.

110

Organometallic gold(III) and gold(I) complexes as catalysts for the 1,3-dipolar cycloaddition to nitrones: synthesis of novel gold-nitrone derivatives, Ade, A.; Cerrada, E.; Contel, M.; Laguna, M.; Merino, P.; Tejero, T. J. Organomet. Chem. 2004, 689, 1788-1795.

109

A comparative study of the stereoselective addition of trimethylsilyl cyanide and diethylaluminum cyanide to chiral cyclic nitrones, Merino, P.; Tejero, T.; Revuelta, J.; Romero, P.; Cicchi, S.; Mannucci, V.; Brandi, A.; Goti, A. Tetrahedron: Asymmetry 2003, 14, 367-379.

108

An investigation of the Lewis acid mediated 1,3-dipolar cycloaddition between N-benzyl-C-(2-pyridyl)nitrone and allylic alcohol. Direct entry to isoxazolidinyl C-nucleosides, Merino, P.; Tejero, T.; Laguna, M.; Cerrada, E.; Moreno, A.; Lopez, J. A. Org. Biomol. Chem. 2003, 1, 2336-2342.

107

A DFT study on the 1,3-dipolar cycloaddition reactions of C-(methoxycarbonyl)-N-methyl nitrone with methyl acrylate and vinyl acetate, Merino, P.; Revuelta, J.; Tejero, T.; Chiacchio, U.; Rescifina, A.; Romeo, G. Tetrahedron 2003, 59, 3581-3592.

106

1,3-Dipolar cycloaddition between N-benzyl-C-glycosyl nitrones and methyl acrylate en route to glycosyl pyrrolidines, Merino, P.; Franco, S.; Merchan, F. L.; Romero, P.; Tejero, T.; Uriel, S. Tetrahedron: Asymmetry 2003, 14, 3731-3743.

105

Stereoselective synthesis of (-)-deacetylanisomycin, Merino, P.; Franco, S.; Lafuente, D.; Merchan, F.; Revuelta, J.; Tejero, T. Eur. J. Org. Chem. 2003, 2877-2881.

104

Nucleophilic additions to nitrones: An alternative gateway to isoxazolidines, pyrrolidines and related compounds. In Targets in Heterocyclic Systems, Merino, P., Attanasi, O.; Spinelli, D., Eds. RSC Publishing: London, 2003; Vol. 7, pp 140-156.

103

Iterative organometallic addition to chiral hydroxylated cyclic nitrones: highly stereoselective syntheses of alpha,alpha'- and alpha,alpha-substituted hydroxypyrrolidines, Goti, A.; Cicchi, S.; Mannucci, V.; Cardona, F.; Guarna, F.; Merino, P.; Tejero, T. Org. Lett. 2003, 5, 4235-4238.

102

Isoxazolidine analogs of pseudouridine: a new class of modified nucleosides, Chiacchio, U.; Corsaro, A.; Mates, J.; Merino, P.; Piperno, A.; Rescifina, A.; Romeo, G.; Romeo, R.; Tejero, T. Tetrahedron 2003, 59, 4733-4738.

101

Enantioselective synthesis of N,O-psiconucleosides, Chiacchio, U.; Borrello, L.; Iannazzo, D.; Merino, P.; Piperno, A.; Rescifina, A.; Richichi, B.; Romeo, G. Tetrahedron: Asymmetry 2003, 14, 2419-2425.

100

Enantioselective synthesis of 4-hydroxy-D-pyroglutamic acid derivatives by an asymmetric 1,3-dipolar cycloaddition, Merino, P.; Revuelta, J.; Tejero, T.; Chiacchio, U.; Rescifina, A.; Piperno, A.; Romeo, G. Tetrahedron: Asymmetry 2002, 13, 167-172.

99

Experimental and theoretical study of the 1,3-dipolar cycloaddition between D-glyceraldehyde nitrones and acrylates. diastereoselective approach to 4-hydroxy pyroglutamic acid derivatives, Merino, P.; Mates, J. A.; Revuelta, J.; Tejero, T.; Chiacchio, U.; Romeo, G.; Iannazzo, D.; Romeo, R. Tetrahedron: Asymmetry 2002, 13, 173-190.

98

Efficient synthesis of (2R,3S)- and (2S,3S)-2-amino-1,3,4-butanetriols through stereodivergent hydroxymethylation of D-glyceraldehyde nitrones, Merino, P.; Franco, S.; Merchan, F. L.; Revuelta, J.; Tejero, T. Tetrahedron Lett. 2002, 43, 459-462.

97

Understanding the High Diastereofacial Discrimination in Nucleophilic Additions to Nitrones. The First Ab Initio Study on the Nucleophilic Addition Reactions of Chiral Nitrones with Grignard Reagents, Merino, P.; Tejero, T. Tetrahedron 2001, 57, 8125-8128.

96

Facial selectivity in the addition of ketene acetals to nitrones towards chiral non-racemic isoxazolidin-5-ones. A semiempirical study, Merino, P.; Mates, J. A. Arkivoc 2001, 12-30.

95

Crystal and molecular structures of N-benzyl-C-(2-pyridyl)nitrone and its ZnBr2 complex. A study of their reactivity, Merino, P.; Anoro, S.; Cerrada, E.; Laguna, M.; Moreno, A.; Tejero, T. Molecules 2001, 6, 208-220.

94

Nucleophilic additions to chiral nitrones: new approaches to nitrogenated compounds, Merino, P.; Franco, S.; Merchan, F. L.; Tejero, T. Synlett 2000, 442-454.

93

Stereodivergent Approaches to the Synthesis of Isoxazolidine Analogues of a-Amino Acid Nucleosides. Total Synthesis of Isoxazolidinyl Deoxypolyoxin C and Uracil Polyoxin C, Merino, P.; Franco, S.; Merchan, F. L.; Tejero, T. J. Org. Chem. 2000, 65, 5575-5589.

92

Stereoselective synthesis of L-isoxazolidinyl thymidine from N-benzyl-1,2-di-O-isopropylidene-D-glyceraldehyde nitrone (BIGN), Merino, P.; Del Alamo, E. M.; Franco, S.; Merchan, F. L.; Simon, A.; Tejero, T. Tetrahedron: Asymmetry 2000, 11, 1543-1554.

91

1,3-Dipolar cycloadditions of N-benzyl furfuryl nitrones with electron-rich alkenes, Merino, P.; Anoro, S.; Merchan, F. L.; Tejero, T. Molecules 2000, 5, 132-152.

90

1,3-Dipolar cycloaddition between hetaryl nitrones and methyl acrylate: Theoretical study and application to the synthesis of functionalized pyrrolidines, Merino, P.; Anoro, S.; Merchan, F.; Tejero, T. Heterocycles 2000, 53, 861-876.

89

1,3-Dipolar Cycloaddition of Furfuryl Nitrones with Acrylates. A Convenient Approach to Protected 4-Hydroxypyroglutamic Acids, Merino, P.; Anoro, S.; Franco, S.; Merchan, F. L.; Tejero, T.; Tunon, V. J. Org. Chem. 2000, 65, 1590-1596.

88

A general method for the vinylation of nitrones. Synthesis of allylhydroxylamines and allylamines, Merino, P.; Anoro, S.; Franco, S.; Gascon, J. M.; Martin, V.; Merchan, F. L.; Revuelta, J.; Tejero, T.; Tunon, V. Synth. Comm. 2000, 30, 2989-3021.

87

Lewis acid stereocontrolled additions of a silyl ketene acetal to 2,3-di-O-isopropylidene-D-glyceraldehyde nitrones. Synthesis of L-isoxazolidinyl nucleosides, Merino, P.; Alamo, E. M. d.; Bona, M.; Franco, S.; Merchan, F. L.; Tejero, T.; Vieceli, O. Tetrahedron Lett. 2000, 41, 9239-9243.

86

Stereochemistry of a-(tert-butoxycarbonylamino) hydroxylamines: 1H NMR analysis of hydroxylamines derived from 2-pyrrolidinyl nitrones, Merino, P.; Franco, S.; Gascon, J. M.; Merchan, F. L.; Tejero, T. Tetrahedron: Asymmetry 1999, 10, 1861-1865.

85

Highly diastereoselective nucleophilic addition of organometallic reagents to 2-pyrrolidinyl nitrones: a semiempirical approach, Merino, P.; Franco, S.; Gascon, J. M.; Merchan, F. L.; Tejero, T. Tetrahedron: Asymmetry 1999, 10, 1867-1871.

84

Chiral hydroxylamines. V. (2S,3S)-N-benzyl-N-[3-(tert-butoxycarbonylamino)-2-butyl]hydroxylamine, Merino, P.; Merchan, F. L.; Tejero, T.; Lanaspa, A. Acta Crystallographica, Section C: Crystal Structure Communications 1998, C54, 85-86.

83

Crystal Structure of methyl (2R,3S,4R)-N-Acetyl-2-amino-5-O-tertbutyldimethylsilyl-3,4-O-isopropylidene-3,4,5-trihydroxypentanoate, Merino, P.; Merchan, F. L.; Tejero, T.; Franco, S. Zeits. Krist. 1998, 213, 135-136.

82

Structures of chiral hydroxylamines. VI. (3R,4S)-N-benzyl-4,5-dihydroxy-3-(hydroxyamino)-4,5-O-isopropylidene-1-pentyne, Merino, P.; Merchan, F. L.; Tejero, T.; Franco, S. Acta Crystallographica, Section C: Crystal Structure Communications 1998, C54, 1003-1004.

81

Totally stereocontrolled synthesis of a,b-diamino acids by addition of Grignard reagents to nitrones derived from L-serine, Merino, P.; Lanaspa, A.; Merchan, F. L.; Tejero, T. Tetrahedron: Asymmetry 1998, 9, 629-646.

80

Nucleophilic Additions of 2-Furyllithium to Carbonyl Derivatives of L-Serine. Formal Synthesis of (2R,3R)-α-Hydroxy Aspartic Acid, Merino, P.; Franco, S.; Merchan, F. L.; Tejero, T. Molecules 1998, 3, 26-30.

79

Crystal Structure of 1-(tert-Butoxycarbonylamino)-1-deoxy-2,3-O-isoprop-ylidene-1-(2-thiazolyl)-D-threo-triitol, Merino, P.; Franco, S.; Merchan, F. L.; Tejero, T. Zeits. Krist. 1998, 213, 133-134.

78

Asymmetric Addition Reactions of Lithium (Trimethylsilyl)acetylide with Chiral a-Amino Nitrones. Synthesis of Diastereomerically Pure N-Hydroxy-a-amino Acids, Merino, P.; Franco, S.; Merchan, F. L.; Tejero, T. J. Org. Chem. 1998, 63, 5627-5630.

77

Asymmetric synthesis of an isoxazolidine nucleoside analog of thymine polyoxin C, Merino, P.; Franco, S.; Merchan, F. L.; Tejero, T. Tetrahedron Lett. 1998, 39, 6411-6414.

76

Synthesis of isoxazolidin-5-ones via stereocontrolled Michael additions of benzylhydroxylamine to L-serine derived a,b-unsaturated esters, Merino, P.; Franco, S.; Merchan, F. L.; Tejero, T. Tetrahedron: Asymmetry 1998, 9, 3945-3949.

75

Modified nucleosides from nitrones: a new and efficient stereoselective approach to isoxazolidinyl thymidine derivatives, Merino, P.; Franco, S.; Garces, N.; Merchan, F. L.; Tejero, T. Chem. Commun. 1998, 493-494.

74

Enantiodivergent Approach to D- and L-Secondary N-Hydroxy-a-amino Acids by Using N-Benzyl-2,3-O-isopropylidene-D-glyceraldehyde Nitrone as an Effective N-Hydroxyglycine Cation Equivalent, Merino, P.; Castillo, E.; Franco, S.; Merchan, F. L.; Tejero, T. J. Org. Chem. 1998, 63, 2371-2374.

73

Ready access to enantiopure 5-substituted-3-pyrrolin-2-ones from N-benzyl-2,3-O-isopropylidene-D-glyceraldehyde nitrone (BIGN), Merino, P.; Castillo, E.; Franco, S.; Merchan, F. L.; Tejero, T. Tetrahedron: Asymmetry 1998, 9, 1759-1769.

72

Nucleophilic additions of Grignard reagents to N-benzyl-2,3-O-isopropylidene-D-glyceraldehyde nitrone (BIGN). Synthesis of (2S,3R) and (2S,3S)-3-phenylisoserine, Merino, P.; Castillo, E.; Franco, S.; Merchan, F. L.; Tejero, T. Tetrahedron 1998, 54, 12301-12322.

71

1,3-Dipolar cycloaddition of C-(2-thiazolyl)nitrones to chiral acrylates. Synthesis of enantiopure a-amino-2-alkylthiazoles and 5-formylpyrrolidin-2-ones, Tejero, T.; Dondoni, A.; Rojo, I.; Merchan, F. L.; Merino, P. Tetrahedron 1997, 53, 3301-3318.

70

Chiral hydroxylamines. IV. 1-(N-benzyl-N-hydroxyamino)-2:3;4:5-di-O-isopropylidene-a-D-mannofuranose, Merino, P.; Merchan, F. L.; Tejero, T.; Franco, S. Acta Crystallographica, Section C: Crystal Structure Communications 1997, C53, 1703-1705.

69

Crystal Structure of (1R,2S)-N-Benzyl-N-[2-(tert-butoxycarbonylamino)-1-(furan-2-yl)-1-propyl]hydroxylamine, Merino, P.; Lanaspa, A.; Merchan, F. L.; Tejero, T. Zeits. Krist. 1997, 212, 323-324.

68

Stereocontrolled synthesis of 2,3-diaminobutanoic acids, Merino, P.; Lanaspa, A.; Merchan, F. L.; Tejero, T. Tetrahedron Lett. 1997, 38, 1813-1816.

67

Stereoselective Grignard reactions to a-amino nitrones. Synthesis of optically active a-aminohydroxylamines and 1,2-diamines, Merino, P.; Lanaspa, A.; Merchan, F. L.; Tejero, T. Tetrahedron: Asymmetry 1997, 8, 2381-2401.

66

A Facile Synthesis of Glycosyl Hydroxylamines, Merino, P.; Franco, S.; Merchan, F. L.; Tejero, T. Synth. Commun. 1997, 27, 3529-3537.

65

Diastereoselective nucleophilic addition of acetylide to N-benzyl-2, 3-O-isopropylidene-D-glyceraldehyde nitrone (BIGN). Stereodivergent synthesis of b-hydroxy-a-(hydroxyamino)- and b-hydroxy-a-amino acids, Merino, P.; Franco, S.; Merchan, F. L.; Tejero, T. Tetrahedron: Asymmetry 1997, 8, 3489-3496.

64

Crystal Structure of 2-Acetamido-1-O-acetyl-2-deoxy-3,4:5,6-di-O-isopropylidene-D-mannitol, Merino, P.; Franco, S.; Junquera, F.; Merchan, F. L.; Tejero, T. Zeits. Krist. 1997, 212, 321-322.

63

Crystal Structure of (2S*,3R*)-N-Benzyl-2-(benzyloxy)-3-(hydroxylamino) butane, Merino, P.; Castillo, E.; Merchan, F. L.; Tejero, T. Zeits. Krist. 1997, 212, 443-444.

62

Crystal Structure of (2S*,3R*)-N-Benzyl-2-(benzyloxy)-3-(hydroxylamino) propane, Merino, P.; Castillo, E.; Merchan, F. L.; Tejero, T. Zeits. Krist. 1997, 212, 441-442.

61

Stereocontrolled addition of Grignard reagents to a-alkoxy nitrones. Synthesis of syn- and anti-3-amino-1,2-diols, Merino, P.; Castillo, E.; Merchan, F. L.; Tejero, T. Tetrahedron: Asymmetry 1997, 8, 1725-1729.

60

A new entry to glycosylamines, Merchan, F. L.; Merino, P.; Tejero, T. Glycoconjugate J. 1997, 14, 497-499.

59

Novel five- and six- membered bisheterocyclic systems from dithiocarbamates and related compounds, Franco, S.; Merchan, F. L.; Merino, P.; Tejero, T. Trends in Heterocyclic Chemistry 1997, 5, 57-74.

58

Stereoselective Addition of 2-Furyllithium and 2-Thiazolyllithium to Sugar Nitrones. Synthesis of Carbon-Linked Glycoglycines, Dondoni, A.; Junquera, F.; Merchan, F. L.; Merino, P.; Scherrmann, M.-C.; Tejero, T. J. Org. Chem. 1997, 62, 5484-5496.

57

Applications of Sugar Nitrones in Synthesis: The Total Synthesis of (+)-Polyoxin J, Dondoni, A.; Franco, S.; Junquera, F.; Merchan, F. L.; Merino, P.; Tejero, T. J. Org. Chem. 1997, 62, 5497-5507.

56

Absolute configuration determination in furfuryl amines and hydroxylamines by circular dichroism, Tejero, T.; Franco, S.; Junquera, F.; Lanaspa, A.; Merchan, F. L.; Merino, P.; Rojo, I. Tetrahedron: Asymmetry 1996, 7, 1529-1534.

55

Structures of chiral nitrones. II. (Z)-N-[(2S)-2-(tert-butoxycarbonylamino)propylidene]benzylamine N-oxide, Merino, P.; Merchan, F. L.; Tejero, T.; Lanaspa, A. Acta Crystallographica, Section C: Crystal Structure Communications 1996, C52, 218-219.

54

Chiral hydroxylamines. II. (1R,2R)-N-benzyl-N-[(3-tert-butoxycarbonyl-2,2-dimethyloxazol-4-yl)(furan-2-yl)methyl]hydroxylamine, Merino, P.; Merchan, F. L.; Tejero, T.; Lanaspa, A. Acta Crystallographica, Section C: Crystal Structure Communications 1996, C52, 2536-2538.

53

Diastereoselective Hydrocyanation of Chiral Nitrones. Synthesis of novel α-(hydroxyamino) nitriles, Merino, P.; LAnaspa, A.; Merchan, F. L.; Tejero, T. J. Org. Chem. 1996, 61, 9028-9032.

52

Chiral hydroxylamines. III. 1-(N-Benzyl-N-hydroxyamino)-1-deoxy-1-(2-furyl)-2,3:4,5-di-O-isopropylidene-L-manno-pentitol, Merino, P.; Junquera, F.; Merchan, F. L.; Tejero, T. Acta Crystallographica, Section C: Crystal Structure Communications 1996, C52, 3197-3198.

51

Direct vinylation and ethynylation of nitrones. Stereodivergent synthesis of allyl and propargyl amines, Merino, P.; Anoro, S.; Castillo, E.; Merchan, F.; Jejero, T. Tetrahedron: Asymmetry 1996, 7, 1887-1890.

50

Enantioselective addition of Grignard reagents to a 2-thiazolyl nitrone, Merchan, F. L.; Merino, P.; Rojo, I.; Tejero, T.; Dondoni, A. Tetrahedron: Asymmetry 1996, 7, 667-670.

49

A straightforward synthesis of L-isoserinal, Junquera, F.; Merchan, F. L.; Merino, P.; Tejero, T. Tetrahedron 1996, 52, 7045-7052.

48

Alkylation of camphor and pinanone imines of 2-(aminomethyl)thiazole. Enantioselective synthesis of 2-(1-aminoalkyl)thiazoles, Dondoni, A.; Merchan, F. L.; Merino, P.; Rojo, I.; Tejero, T. Synthesis 1996, 641-646.

47

(Z)-N-[(2R,3R)-2-(tert-Butoxycarbonylamino)-3-(tert-butyldiphenylsiloxy)butylidene]benzylamine N-oxide, Merino, P.; Merchan, F. L.; Tejero, T.; Lanaspa, A. Acta Crystallographica, Section C: Crystal Structure Communications 1995, C51, 1949-1950.

46

Chiral hydroxylamines. I. 1-(N-benzyl-N-hdyroxyamino)-1-deoxy-2,3-O-isopropylidene-1-(1-methylimidazol-2-yl)-D-threo-triitol, Merino, P.; Merchan, F. L.; Tejero, T. Acta Crystallographica, Section C: Crystal Structure Communications 1995, C51, 2400-2401.

45

Stereoselective addition of cyanide reagents to nitrones, Merchan, F. L.; Merino, P.; Tejero, T. Tetrahedron Lett. 1995, 36, 6949-6952.

44

Determination of the absolute configuration of a-amino-2-alkylthiazoles by circular dichroism, Merchan, F. L.; Merino, P.; Rojo, I.; Tejero, T.; Dondoni, A. Tetrahedron: Asymmetry 1995, 6, 2145-2148.

43

Synthesis of 2,2'-(alkylenediamino)dibenzazoles: New heterocyclic tetradentate ligands, Melendez, E.; Merchan, F. L.; Tejero, T.; Merino, P.; Garcia, M. An. Quim. 1995, 90, 487-490.

42

An improved synthesis of ketonitrones, Franco, S.; Merchan, F. L.; Merino, P.; Tejero, T. Synth. Commun. 1995, 25, 2275-2284.

41

Chelation- and Non-chelation-Controlled Addition of 2-(Trimethylsilyl)thiazole to a-Amino Aldehydes: Stereoselective Synthesis of the b-Amino-a-hydroxy Aldehyde Intermediate for the Preparation of the Human Immunodeficiency Virus Proteinase Inhibitor Ro 31-8959, Dondoni, A.; Perrone, D.; Merino, P. J. Org. Chem. 1995, 60, 8074-8080.

40

Total synthesis of (+)-polyoxin J, Dondoni, A.; Junquera, F.; Merchan, F. L.; Merino, P.; Tejero, T. Chem. Commun. 1995, 2127-2128.

39

Stereoselective homologation-amination of aldehydes by addition of their nitrones to C-2 metalated thiazoles - a general entry to a-amino aldehydes and amino sugars, Dondoni, A.; Franco, S.; Junquera, F.; Merchan, F. L.; Merino, P.; Tejero, T.; Bertolasi, V. Chem. Eur. J. 1995, 1, 505-520.

38

Tunable stereoselectivity in the addition of 2-lithiothiazole to L-serinal derived N-benzyl nitrone. Synthesis of C-2 epimer 2,3-diamino-4-hydroxybutanals, Dondoni, A.; Merchan, F. L.; Merino, P.; Tejero, T.; Bertolasi, V. Chem. Commun. 1994, 1731-1733.

37

Nitrones in Organic Synthesis. Synthesis of Secondary Allyl Amines, Dondoni, A.; Merchan, F.; Merino, P.; Tejero, T. Synth. Commun. 1994, 24, 2551-2555.

36

Installation of the Pyruvate Unit in Glycidic Aldehydes via a Wittig Olefination-Michael Addition Sequence Utilizing a Thiazole-Armed Carbonyl Ylide. A New Stereoselective Route to 3-Deoxy-2-Ulosonic Acids and the Total Synthesis of DAH, KDN, and 4-epi-KDN, Dondoni, A.; Marra, A.; Merino, P. J. Am. Chem. Soc. 1994, 116, 3324-3336.

35

Addition of 2-Lithiofuran to Chiral alpha-Alkoxy Nitrones. A Stereoselective Approach to alpha-epimer-beta-alokoxy-alfa aminoacids, Dondoni, A.; Junquera, F.; Merchan, F. L.; Merino, P.; Tejero, T. Synthesis 1994, 1450-1455.

34

Total synthesis of thymine polyoxin C, Dondoni, A.; Junquera, F.; Merchan, F. L.; Merino, P.; Tejero, T. Tetrahedron Lett. 1994, 35, 9439-9442.

33

Stereo-controlled homologation of 1,2:3,4-di-O-isopropylidene-a-D-galacto-hexodialdo-1,5-pyranose to 7-deoxynonodialdose epimers via thiazole-aldehyde synthesis, Dondoni, A.; Ianelli, S.; Kniezo, L.; Merino, P.; Nardelli, M. J. Chem. Soc., Perkin Trans. 1 1994, 1231-1239.

32

Synthesis of N-Benzyl Nitrones, Dondoni, A.; Franco, S.; Junquera, F.; Merchan, F. L.; Merino, P.; Tejero, T. Synth. Commun. 1994, 24, 2537-2550.

31

Total chemical synthesis of aza sugars via thiazole intermediates. Stereodivergent routes to (-)-nojirimycin, (-)-mannojirimycin and their 3-deoxy derivatives from serine, Dondoni, A.; Merino, P.; Perrone, D. Tetrahedron 1993, 49, 2939-2956.

30

Two-carbon chain extension of chiral aldehydes via 2-alkenylthiazoles: synthesis of g-functionalized alkanals, Dondoni, A.; Merino, P.; Orduna, J.; Perrone, D. Synthesis 1993, 277-279.

29

Iterative methodology for the stereocontrolled synthesis of polyol chains employing 2-acetylthiazole as lactaldehyde equivalent, Dondoni, A.; Merino, P. Synthesis 1993, 903-908.

28

Diastereoselective homologation of D-(R)-glyceraldehyde acetonide using 2-(trimethylsilyl)thiazole: 2-O-benzyl-3,4-isopropylidene-D-erythrose (1,3-dioxolane-4-acetaldehyde, 2,2-dimethyl-a-(phenylmethoxy)-, [R-(R*,R*)]-), Dondoni, A.; Merino, P. Org. Synth. 1993, 72, 21-31.

27

Stereocontrol by diethylaluminum chloride in the addition of 2-lithiofuran and N-methyl-2-lithioimidazole to a-alkoxy nitrones. Total synthesis of 5-O-carbamoylpolyoxamic acid, Dondoni, A.; Franco, S.; Merchan, F. L.; Merino, P.; Tejero, T. Tetrahedron Lett. 1993, 34, 5479-5482.

26

Stereocontrolled addition of 2-lithiothiazole to the nitrone derived from D-glyceraldehyde acetonide. A revision and extension, Dondoni, A.; Franco, S.; Merchan, F. L.; Merino, P.; Tejero, T. Tetrahedron Lett. 1993, 34, 5475-5478.

25

Stereocontrolled addition of 2-thiazolyl organometallic reagents to C-galactopyranosylnitrone. A formal synthesis of destomic acid and lincosamine, Dondoni, A.; Franco, S.; Merchan, F.; Merino, P.; Tejero, T. Synlett 1993, 78-80.

24

Construction of all O-alkoxy D-tetrose and D-pentose stereoisomers from 2,3-O-isopropylidene-D-glyceraldehyde using 2-(trimethylsilyl)thiazole as a formyl anion equivalent, Dondoni, A.; Orduna, J.; Merino, P. Synthesis 1992, 201-210.

23

4-O-Benzyl-2,3-O-isopropylidene-D-erythrose and -D-threose from 2,3-O-isopropylidene-D-glyceraldehyde via thiazole intermediates. Synthesis of 2-deoxykanosamine, Dondoni, A.; Merino, P. Synthesis 1992, 196-200.

22

Stereoselective aminohomologation of chiral a-alkoxy aldehydes via thiazole addition to nitrones. Application to the synthesis of N-acetyl-D-mannosamine, Dondoni, A.; Junquera, F.; Merchan, F. L.; Merino, P.; Tejero, T. Tetrahedron Lett. 1992, 33, 4221-4224.

21

Diheterocyclic compounds from dithiocarbamates and derivatives thereof. VI. Unsymmetrical N1,N4-bis(2-benzazolyl)sulfanilamides, Melendez, E.; Merchan, F. L.; Merino, P.; Orduna, J.; Urchegui, R. J. Het. Chem. 1991, 28, 653-656.

20

The reaction of anthranilic acid with thionyl chloride: the actual structure of Kametani's sulfinamide anhydride, Garin, J.; Merino, P.; Orduna, J.; Tejero, T.; Uriel, S. Tetrahedron Lett. 1991, 32, 3263-3264.

19

Synthesis of unsymmetrical diheteroarylbenzenes: benzazole and quinazoline derivatives, Garin, J.; Melendez, E.; Merchan, F. L.; Merino, P.; Orduna, J.; Tejero, T. J. Het. Chem. 1991, 28, 359-363.

18

Homologation of L-threonine to a-epimer b-amino-a,g-dihydroxy aldehydes and acids via stereoselective reduction of 2-thiazolyl amino ketones, Dondoni, A.; Perrone, D.; Merino, P. Chem. Commun. 1991, 1313-1314.

17

Stereocontrolled total synthesis of galactostatin from serine, Dondoni, A.; Merino, P.; Perrone, D. Chem. Commun. 1991, 1576-1578.

16

Stereoselective construction of polyhydroxyalkyl 2-triazolyl ketones (thiazole ketoses) from D-glyceraldehyde and D-arabinose acetonides by Wittig-Michael sequence. A route to D-gluco-KDO, Dondoni, A.; Merino, P.; Orduna, J. Tetrahedron Lett. 1991, 32, 3247-3250.

15

Chemistry of the enolates of 2-acetylthiazole: aldol reactions with chiral aldehydes to give 3-deoxy aldos-2-uloses and 3-deoxy 2-ulosonic acids. A short total synthesis of 3-deoxy-D-manno-2-octulosonic acid (KDO), Dondoni, A.; Merino, P. J. Org. Chem. 1991, 56, 5294-5301.

14

Diheterocyclic compounds from dithiocarbamates and derivatives thereof. V. 4,4'-Dioxo-2,2'-dithioxo(dioxo)-6,6'-biquinazolines, Garin, J.; Melendez, E.; Merchan, F. L.; Merino, P.; Orduna, J.; Tejero, T.; Vinegra, M. J. Het. Chem. 1990, 27, 1351-1354.

13

Chemoselectivity in The Oxidation of Unsymmetrical Thioureas with NBS/Sulfuric Acid: Benzothiazoles vs. 1,2,4-Thiadiazoles, Garin, J.; Melendez, E.; Merchan, F. L.; Merino, P.; Orduna, J.; Tejero, T. Synth. Commun. 1990, 20, 2324-2327.

12

Diheterocyclic compounds from dithiocarbamates and derivatives thereof. II. 2,2'-Diamino-6,6'-bibenzoazoles, Garin, J.; Melendez, E.; Merchan, F. L.; Merino, P.; Orduna, J.; Tejero, T. J. Het. Chem. 1990, 27, 321-326.

11

Diheterocyclic compounds from dithiocarbamates and derivatives thereof. III. 3,3'-Arylenebis(2,4-dioxo-1,2,3,4-tetrahydroquinazolines), Garin, J.; Melendez, E.; Merchan, F. L.; Merino, P.; Orduna, J.; Tejero, T. J. Het. Chem. 1990, 27, 1341-1344.

10

Diheterocyclic compounds from dithiocarbamates and derivatives thereof. IV. 3,3'-Arylenebis(4-oxo-2-thioxo-1,2,3,4-tetrahydroquinazolines), Garin, J.; Melendez, E.; Merchan, F. L.; Merino, P.; Orduna, J.; Tejero, T. J. Het. Chem. 1990, 27, 1345-1349.

9

Diheterocyclic compounds from dithiocarbamates and derivatives thereof. I. 2,2'-(Arylenediamino)bisbenzoazoles, 2,2'-(arylenediamino)bis(imidazopyridines) and 8,8'-(arylenediamino)bispurines, Garin, J.; Melendez, E.; Merchan, F. L.; Merino, P.; Orduna, J.; Tejedor, R.; Tejero, T. J. Het. Chem. 1990, 27, 221-226.

8

A divergent route to nojirimycin analogs from L-serinal and 2-acetylthiazole, Dondoni, A.; Fantin, G.; Fogagnolo, M.; Merino, P. Chem. Commun. 1990, 854-856.

7

A concise new route to 3-deoxy-D-manno-2-octulosonic acid (KDO) from D-arabinose and 2-acetylthiazole, Dondoni, A.; Fantin, G.; Fogagnolo, M.; Merino, P. Tetrahedron Lett. 1990, 31, 4513-4516.

6

Chain-elongation of dialdoses containing the a-galactopyranosyl group by a Wittig reaction with 2-thiazolylmethylenetriphenylphosphorane. The thiazole route to long-chain alkene sugars, Dondoni, A.; Fantin, G.; Fogagnolo, M.; Merino, P. J. Carbohydr. Chem. 1990, 9, 735-744.

5

Regio- and stereoselective conjugate addition of nitrogen nucleophiles to 2-alkenyl-N-methylthiazolium iodides. Synthesis of D-3-epi-daunosamine and some lincosamine analogs, Dondoni, A.; Fantin, G.; Fogagnolo, M.; Merino, P. Tetrahedron 1990, 46, 6167-6184.

4

A Facile New Method For The Preparation of Aromatic Diisothiocyanates, Garin, J.; Melendez, E.; Merchan, F. L.; Merino, P.; Tejero, T. Bull. Soc. Chim. Belg. 1989, 98, 289-290.

3

Tetramethyl Bis[N-(2-Benzothiazolyl) Dithiocarbon-Imidates]: Novel Reagents For Heterocyclic Polymer Synthesis, Garin, J.; Melendez, E.; Merchan, F. L.; Merino, P.; Orduna, J.; Tejero, T. Synth. Commun. 1989, 19, 2389-2399.

2

On The Reaction of Aromatic Amines with Carbon Disulfide: A Facile Modified Preparation of Bis(Dithiocarbamic) Acid Derivatives, Garin, J.; Melendez, E.; Merchan, F. L.; Merino, P.; Tejero, T. Bull. Soc. Chim. Belg. 1988, 97, 791-792.

1

Dithiocarbamoyl Derivatives: Useful Reagents In Heterocyclic Synthesis, Garin, J.; Melendez, E.; Merchan, F.; Merino, P.; Orduna, J.; Tejero, T. Il Farmaco 1988, 437, 1183-1194.

 

Reviews

32

Direct Hydroxymethylation of C=N Double Bonds
Lett. Org. Chem. 2018, . DOI:


31

New Mechanistic Interpretation for Nitrone Reactivity
Org. Biomol. Chem.
. 2017, 15, 3355-3530. DOI: 10.1039/c7ob00429u

30

Chemical Approaches to Inhibitors of Isoprenoid Biosynthesis: Targeting Farnesyl and Geranylgeranyl Pyrophosphate Synthases, RSC. Adv. 2017, 7, 10947-10967. DOI: 10.1039/c6ra28316k

29

Nucleoside Diphosphate Sugar Analogues that Target Glycosyltransferases,
Asian
J. Org. Chem.. 2016, 1413-1427. DOI: 10.1002/ajoc.201600396

28

Design and Synthesis of Dopaminergic Agonists, Matute, M. S.; Matute, R.; Merino, P. Curr. Med. Chem. 2016, 23.
DOI: 10.2174/0929867323666160504103621 

27

Recent Advances on Asymmetric Nitroso Aldol Reaction, Merino, P.; Tejero, T.; Delso, I.; Matute, R. Synthesis 2016, 48, 653-676.

26

Recent advances in the preparation of enantiomerically pure hydroxylamines from nitrones, Matute, R.; Garcia-Viñuales, S.; Hayes, H.; Ghirardello, M.; Daru, A.; Tejero, T.; Delso, I.; Merino, P. Curr. Org. Synth. 2016, 13, 669-686

25

Oxidation reactions of Furan, Merino, P. Org. React. 2015, 87, 1-256.

24

Recent   Advances   on   the   Enantioselective   Synthesis   of   C-Nucleosides Inhibitors of Inosine Monophosphate Dehydrogenase (IMPDH), Merino, P.; Ghirardello, M.; Tejero, T.; Delso, I.; Matute, R. Curr. Top. Med. Chem. 2014, 14, 1212-1224.

23

Biosynthetic Pathways to Glycosidase Inhibitors, Gomollón-Bel, F.; Delso, I.; Tejero, T.; Merino, P. Curr. Chem. Biol. 2014, 8, 10-16.

22

Cross-coupling reactions for the synthesis of C-glycosides and related compounds, Merino, P.; Tejero, T.; Marca, E.; Gomollon-Bel, F.; Delso, I.; Matute, R. Heterocycles 2012, 86, 791-820.

21

Recent advances on the synthesis of piperidines through ruthenium-catalyzed ring-closing metathesis (RCM) reactions, Merino, P.; Tejero, T.; Greco, G.; Marca, E.; Delso, I.; Gómez-SanJuan, A.; Matute, R. Heterocycles 2012, 84, 75-100.

20

Recent progress on fucosyltransferase inhibitors, Merino, P.; Tejero, T.; Delso, I.; Hurtado-Guerrero, R.; Gomez-SanJuan, A.; Sadaba, D. Mini-Rev. Med. Chem. 2012, 12, 1455-1464.

19

Chemical synthesis of five-membered nitrogen heterocycles by reductive cyclization methods, Tejero, T.; Merino, P.; Delso, I.; Sadaba, D. Targets Heterocycl. Syst. 2011, 15, 164-192.

18

Mannich-type reactions with Nitrones, Oximes and Hydrazones, Merino, P.; Tejero, T. Synlett 2011, 1965-1977.

17

Organocatalytic activation of imines and related compounds through hydrogen-bond interactions, Merino, P.; Delso, I.; Tejero, T.; Roca-Lopez, D.; Isas, A.; Matute, R. Curr. Org. Chem.2011, 15, 2184-2209.

16

Chemical Synthesis of Heterocyclic-Sugar Nucleoside Analogues, Romeo, G.; Chiacchio, U.; Corsaro, A.; Merino, P. Chem. Rev. 2010, 110, 3337-3370.

15

Recent developments on rotaxane-based shuttles, Rescifina, A.; Zagni, C.; Iannazzo, D.; Merino, P. Curr. Org. Chem. 2009, 13, 448-481.

14

Chemistry and biology of imino-sugar di- and oligosaccharides, Merino, P.; Delso, I.; Marca, E.; Tejero, T.; Matute, R. Curr. Chem. Biol. 2009, 3, 253-271.

13

Concerted molecular rearrangements. In Seminars in Organic Synthesis, "A. Corbella" Summer School, 34th, Garnano, Italy, June 22-26, 2009, Merino, P., 2009; pp 73-96.

12

Catalytic Enantioselective Aza-Henry Reactions, Marques-Lopez, E.; Merino, P.; Tejero, T.; Herrera, R. P. Eur. J. Org. Chem. 2009, 2401-2420.

11

The role of the indole in important organocatalytic enantioselective Friedel-Crafts alkylation reactions, Marques-Lopez, E.; Diez-Martinez, A.; Merino, P.; Herrera, R. P. Current Organic Chemistry 2009, 13, 1585-1609.

10

Current developments in the synthesis and biological activity of aza-C-nucleosides: immucillins and related compounds, Merino, P.; Tejero, T.; Delso, I. Curr. Med. Chem. 2008, 15, 954-967.

9

Furan oxidations in organic synthesis. Recent advances and applications, Merino, P.; Tejero, T.; Delso, J. I.; Matute, R. Curr.Org. Chemistr. 2007, 11, 1076-1091.

8

Heterocyclic nucleosides: chemical synthesis and biological properties, Merino, P. Curr. Med. Chem. 2006, 13, 539-545.

7

Stereoselective allylation and vinylation reactions of imines and related compounds, Merino, P.; Tejero, T.; Delso, J. I.; Mannucci, V. Curr. Org. Synth. 2005, 2, 479-498.

6

New developments in nucleophilic additions to nitrones, Merino, P. Compt. Rend. Chim. 2005, 8, 775-788.

5

Heterocyclic nucleosides. Chemical synthesis and biological properties, Merino, P. Cur. Med. Chem. 2002, 1, 389-411.

4

Oxidations of furan rings in organic synthesis: Expanding synthetic utility of aromatic heterocycles. In Rec. Res. Dev. Synth. Org. Chem., Merino, P.; Franco, S.; Merchan, F. L.; Tejero, T., Pandalai, S., Ed. 2000; Vol. 3, pp 65-74.

3

Recent developments on chemistry and biological activity of nucleoside analogues with an extra heteroatom in the sugar ring. In Rec. Res. Dev. Org. Chemistry, Merino, P.; Franco, S.; Merchan, F. L.; Tejero, T., Pandalai, S., Ed. 2000; Vol. 4, pp 227-237.

2

Recent advances in the reaction of metalated aromatic heterocycles with carbonyl compounds and their imino derivatives, Merino, P. Progr. Het. Chem. 1999, 11, 21-44.

1

Asymmetric nucleophilic additions to chiral nitrones: Scope and applications. In Rec. Res. Dev Synth Org Chem, Merino, P.; Franco, S.; Merchan, F. L.; Tejero, T., Pandalai, S., Ed. 1998; Vol. 1, pp 109-121.

Book chapters

20 Oxidation reactions of Furan, Merino, P. Org. React. 2015, 87, 1-256.

19

Mannich-type reactions. Merino, P., In Science of Synthesis. C-1 Building Blocks in Organic Synthesis,  Leeuwen, P. W. N. M. v., Ed. Georg Thieme Verlag: Stuttgart, 2014; pp 311-331.

18

CN additions to C=O and C=N bonds. Merino, P., In Comprehensive Organic Synthesis 2nd ed., Knochel, P.; Molander, G. A., Eds. Elsevier: Oxford, 2014; Vol. 1, pp 697-750.

17

Recent advances in the chemical synthesis of aza-nucleosides. Tejero, T.; Delso, I.; Merino, P., In Chemical Synthesis of Nucleoside Analogues, Merino, P., Ed. John Wiley and sons: Hoboken, 2013; pp 699-725.

16

Chemical synthesis of conformationally constrained PNA monomers. Merino, P.; Matute, R., In Chemical Synthesis of Nucleoside Analogues,  Merino, P., Ed. John WIley and sons: Hoboken, 2013; pp 847-880.

15

Nitrones and cyclic analogues. Merino, P., An update. In Science of Synthesis,  Schaumann, E., Ed. George Thieme: Stuttgart, 2011; Vol. 2010/4, pp 325-403.

14

2-(Trimethylsilyl)thiazole, Dondoni, A.; Merino, P.; Sanchez-Sancho, F.; Zarzuelo, M. M.; Garranzo, M. Handbook of Reagents for Organic Synthesis: Reagents for Silicon-Mediated Organic Synthesis 2011, 712-719.

13

Annulated Benzenes (1H-Cyclopropabenzenes, 1,2-Dihydrocyclobutabenzenes, Indanes, and Indenes). Merino, P., In Compounds with All-Carbon Functions. Monocyclic Arenes, Quasiarenes, and Annulenes, Siegel, J. S.; Tobe, Y., Eds. Georg Thieme Verlag: Stuttgart-New York, 2008; Vol. 45a, pp 253-327.

12

Cyclopentadienyl Anions, Cyclopentadienones, and Heteroatom Analogues. Merino, P.,  In Compounds with All-Carbon Functions. Monocyclic Arenes, Quasiarenes, and Annulenes, Siegel, J. S.; Tobe, Y., Eds. Georg Thieme Verlag: Stuttgart-New York, 2008; Vol. 45a, pp 109-156.

11

Cyclopropenium Salts, Cyclopropenones and Heteroatom Analogues, and Cyclopropenyl Radicals and Anions. Merino, P., In Compounds with All-Carbon Functions. Monocyclic Arenes, Quasiarenes, and Annulenes, Siegel, J. S.; Tobe, Y., Eds. Georg Thieme Verlag: Stuttgart-New York, 2008; Vol. 45a, pp 11-48.

10

Acetals OX/OR. Merino, P., In Science of Synthesis, Warriner, S., Ed. George Thieme: Stuttgart, 2007; Vol. 29, pp 707-800.

9

2-(Trimethylsilyl)thiazole - First Update to document cited in CA149:288259, Dondoni, A.; Merino, P.; Sanchez-Sancho, F.; Zarcuelo, M. M.; Garranzo, M. e-EROS Encyclopedia of Reagents for Organic Synthesis 2007, No pp given.

8

Nitrones an its Cyclic Analogues. Merino, P., In Science of Synthesis, Bellus, D.; Padwa, A., Eds. George Thieme: Stuttgart, 2004; Vol. 27, pp 511-580.

7

Benzothiazole, Dondoni, A.; Merino, P. e-EROS Encyclopedia of Reagents for Organic Synthesis 2001, No pp given.

6

2-Methylbenzothiazole, Dondoni, A.; Merino, P. e-EROS Encyclopedia of Reagents for Organic Synthesis 2001, No pp given.

5

2-(Trimethylsilyl)thiazole, Dondoni, A.; Merino, P. e-EROS Encyclopedia of Reagents for Organic Synthesis 2001, No pp given.

4

Thiazoles, Dondoni, A.; Merino, P. Comprehensive Heterocyclic Chemistry II 1996, 3, 373-474.

3

2-(Trimethylsilyl)thiazole. Dondoni, A.; Merino, P., In e-EROS Encyclopedia of Reagents for Organic Synthesis, 1995; pp 5313-5315.

2

2-Methylbenzothiazole. Dondoni, A.; Merino, P., In e-EROS Encyclopedia of Reagents for Organic Synthesis, 1995; pp 3426-3427.

1

Benzothiazole. Dondoni, A.; Merino, P., In e-EROS Encyclopedia of Reagents for Organic Synthesis, 1995; pp 298-300.

 

Edited Books

Chemical Synthesis of Nucleoside Analogues
Pedro Merino (Wiley, ISBN: 978-1-1180-0751-8) \ March 2013. 921 pages
Read more...

Target in Heterocyclic Systems. Vol. 19. 2015
Orazio A. Attanasi, Pedro Merino, Domenico Spinelli
Read more ...


Others

22

Herrera, R. P.; Merino, P. In Uncatalyzed multicomponent synthesis of α-hydrazido phosphonates, Abstracts of Papers, 239th ACS National Meeting, San Francisco, CA, United States, March 21-25, 2010, 2010; pp ORGN-71.

21

¿Por qué no es probable una vida basada en el silicio?, Merino, P. El Esceptico 2006, 82-85.

20

Stereoselective preparation of optically pure methyl 4(R)-N-(tert-butoxycarbonyl)-4-hydroxypyroglutamate, Merino, P.; Franco, S.; Merchan, F.; Revuelta, J.; Tejero, T. International Electronic Conferences on Synthetic Organic Chemistry, 5th, 6th, Sept. 1-30, 2001 and 2002 [and] 7th, 8th, Nov. 1-30, 2003 and 2004 2004, 1268-1273.

19

Professor Enrique Melendez. A tribute, Merino, P. Arkivoc 2004, 1-4.

18

Kappe, O.; Merino, P.; Marzinzik, A.; Wennemers, H.; Wirth, T.; Vanden Eynde, J.-J.; Lin, S.-K. In Proceedings of ECSOC-5. The fifth international electronic conference on synthetic organic chemistry, 2001.

17

Tejero, T.; Anoro, S.; Merchan, F. L.; Merino, P. In 1,3-Dipolar cycloadditions of N-benzyl-C-furfurylnitrones to vinyl ethers and α,β-unsaturated esters, Proceedings. ECSOC-3, Proc. ECSOC-4, 2000; pp 50-58.

16

Crystal and molecular structures of N-benzyl-C-(2-pyridyl) nitrone and its ZnBr2 complex, Merino, P.; Anoro, S.; Tejero, T.; Laguna, M.; Cerrada, E.; Moreno, A. Proceedings of ECSOC-3, [and] Proceedings of ECSOC-4, Sept. 1-30, 1999 and 2000 2000, 502-509.

15

Polyalkoxy nitrones as chiral building blocks in asymmetric synthesis, Merino, P.; Tejero, T. Proceedings of ECSOC-1: The First International Electronic Conference on Synthetic Organic Chemistry; [and] Proceedings of ECSOC-2: The Second International Electronic Conference on Synthetic Organic Chemistry, Sept. 1-30, 1997, 1998 1999, 118-128.

14

Merino, P.; Franco, S.; Merchan, F. L.; Tejero, T. In Nucleophilic additions of 2-furyllithium to carbonyl derivatives of L-serine. Formal synthesis of (2R,3R)-β-hydroxy aspartic acid, Proceedings of ECSOC-1: The First International Electronic Conference on Synthetic Organic Chemistry; [and] Proceedings of ECSOC-2: T, 1999; pp 328-334.

13

(1R,2S)-N-benzyl-N-[(2,2-dimethyl-1,3-dioxolan-4-yl)-(2-benzofuryl)methyl]hydroxylamine, Merino, P.; Franco, S.; Merchan, F. L.; Tejero, T. Molecules [Electronic Publication] 1998, 3, M77.

12

(1S,2S)-N-benzyl-N-[(2,2-dimethyl-1,3-dioxolan-4-yl)-(2-benzofuryl)methyl]hydroxylamine, Merino, P.; Franco, S.; Merchan, F. L.; Tejero, T. Molecules [Electronic Publication] 1998, 3, M78.

11

(1R,2S)-N-benzyl-N-[(2,2-dimethyl-1,3-dioxolan-4-yl)-(2-benzothiazolyl)methyl]hydroxylamine, Merino, P.; Franco, S.; Merchan, F. L.; Tejero, T. Molecules [Electronic Publication] 1998, 3, M79.

10

(1S,2S)-N-benzyl-N-[(2,2-dimethyl-1,3-dioxolan-4-yl)-(2-benzothiazolyl)methyl]hydroxylamine, Merino, P.; Franco, S.; Merchan, F. L.; Tejero, T. Molecules [Electronic Publication] 1998, 3, M80.

9

(1R,2S)-N-benzyl-N-[(2,2-dimethyl-1,3-dioxolan-4-yl)-(2-benzothienyl)methyl]hydroxylamine, Merino, P.; Franco, S.; Merchan, F. L.; Tejero, T. Molecules [Electronic Publication] 1998, 3, M81.

8

(1S,2S)-N-benzyl-N-[(2,2-dimethyl-1,3-dioxolan-4-yl)-(2-benzothienyl)methyl]hydroxylamine, Merino, P.; Franco, S.; Merchan, F. L.; Tejero, T. Molecules [Electronic Publication] 1998, 3, M82.

7

(1S,2S)-N-benzyl-N-[(2,2-dimethyl-1,3-dioxolan-4-yl)-(1-methylimidazol-2-yl)methyl]hydroxylamine, Merino, P.; Franco, S.; Merchan, F. L.; Tejero, T. Molecules [Electronic Publication] 1998, 3, M83.

6

(1R,2S)-N-benzyl-N-[(2,2-dimethyl-1,3-dioxolan-4-yl)-(1-methylimidazol-2-yl)methyl]hydroxylamine, Merino, P.; Franco, S.; Merchan, F. L.; Tejero, T. Molecules [Electronic Publication] 1998, 3, M84.

5

(1R,2S)-N-benzyl-N-[(2,2-dimethyl-1,3-dioxolan-4-yl)-(2-thienyl)methyl]hydroxylamine, Merino, P.; Franco, S.; Merchan, F. L.; Tejero, T. Molecules [Electronic Publication] 1998, 3, M85.

4

(1S,2S)-N-benzyl-N-[(2,2-dimethyl-1,3-dioxolan-4-yl)-(2-thienyl)methyl]hydroxylamine, Merino, P.; Franco, S.; Merchan, F. L.; Tejero, T. Molecules [Electronic Publication] 1998, 3, M86.

3

Stereocontrolled nucleophilic additions of lithiated heterocycles to nitrones. Synthesis and structural characterization of novel chiral (hydroxyamino)methyl heterocycles, Merino, P.; Franco, S.; Martinez, I.; Merchan, F. L.; Tejero, T. ECHET98: Electronic Conference on Heterocyclic Chemistry, June 29-July 24, 1998 1998, 35-40.

2

A short and efficient asymmetric synthesis of 5-substituted Δ3-pyrrolin-2-ones. A new approach to 2-pyrrolidones and pyrrolidines, Merino, P.; Merchan, F.; Tejero, T. Electron. Conf. Heterocycl. Chem., [Proc.] 1997, No pp given.

1

Models for the addition of metalated heterocycles to α-amino nitrones, Lanaspa, A.; Merchan, F. L.; Merino, P.; Tejero, T.; Dondoni, A. Electronic Conference on Trends in Organic Chemistry [CD-ROM] 1996, Paper 9.